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Kinesin Kinesin

Inhibitors

Cat.No.  Name Information
M13687 AZ82 AZ82 is a selective kinesin-like protein KIFC1 (HSET/KIFC1) inhibitor, with a Ki of 43 nM and an IC50 of 300 nM for KIFC1.
M10666 CW069 CW069 is an allosteric inhibitor of HSET with IC50 of 75 μM, it showed marked activity against HSET in vitro.
M9174 ARQ 621 ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor.
M8930 EMD534085 EMD534085 is a potent and selective inhibitor of the mitotic kinesin-5 with an IC50 of 8 nM.
M8918 BAY 1217389 BAY 1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM.
M7876 K-858 Eg5 is a key protein involved in the formation of bipolar spindles.
M5230 Monastrol Monastrol is a cell-permeable small molecule inhibitor of kinesin-5(KIF11) which is essential for maintaining separation of the half-spindles.
M3672 AZD4877 AZD4877 is a synthetic kinesin spindle protein (KSP) inhibitor with potential antineoplastic activity.
M3216 ARRY-520 ARRY-520 is a potent and selective kinesin spindle protein (KSP) inhibitor with an IC50 of 15 nM for A2780, CP70 and 01-28 cell lines in vitro.
M2868 MPI-0479605 MPI-0479605 is an ATP competitive and selective inhibitor of mitotic kinase Mps1 with IC50 of 1.8 nM, >40-fold selectivity over other kinases.
M2171 GSK923295 GSK923295 is an allosteric inhibitor of CENP-E with Ki value of 3.2 nM.
M2128 AZ3146 AZ3146 is a potent and selective monopolar spindle 1 (Mps1) kinase inhibitor with IC50 of 35 nM.
M1983 SB-743921 SB-743921 is a highly potent and active KSP inhibitor with a Ki of 0.1 nM for KSP (Eg5).
M1786 Ispinesib Ispinesib (SB 715992) is the first potent, highly specific small-molecule inhibitor of kinesin spindle protein (KSP) with an IC50 of 4.1 nM.


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