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Litronesib

Cat. No. M30868

All AbMole products are for research use only, cannot be used for human consumption.

Litronesib Structure
Synonym:

LY2523355

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Quality Control & Documentation
Biological Activity

Litronesib (LY2523355) is a selective mitosis-specific kinesin Eg5 inhibitor, with antitumor activity.

Chemical Information
Molecular Weight 511.7
Formula C23H37N5O4S2
CAS Number 910634-41-2
Form Solid
Solubility (25°C) DMSO ≥ 50 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Rinkal Chamariya, et al. Anticancer Agents Med Chem. Role of KSP Inhibitors as Anti-cancer Therapeutics: An Update

[2] Prabhat Pratap Singh Tomar, et al. Viruses. Blockers of the SARS-CoV-2 3a Channel Identified by Targeted Drug Repurposing

[3] Steven W Baertschi, et al. J Pharm Sci. Investigation of the mechanism of racemization of litronesib in aqueous solution: unexpected base-catalyzed inversion of a fully substituted carbon chiral center

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  Catalog
Abmole Inhibitor Catalog




Keywords: Litronesib, LY2523355 supplier, Kinesin, inhibitors, activators

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