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CGRP Receptor Calcitonin gene-related peptide Receptor

Cat.No.  Name Information
M53228 α-CGRP (mouse, rat) α-CGRP (mouse, rat), a neuropeptide (calcitonin gene-related peptide (CGRP)) mainly expressed in neuromuscular junction, is a potent vasodilator.
M40804 Rimegepant Sulfate Rimegepant Sulfate is a potent, selective, competitive, orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki of 0.027 nM.May be used in migraine-related studies.
M40614 Calcitonin (human) Calcitonin (human) is a calcitonin that lowers blood calcium levels and inhibits bone resorption and may be used in studies related to hypercalcemia or osteoporosis.
M28370 Cagrilintide acetate Cagrilintide acetate is an investigational novel long-acting acylated amylin analogue, acts as nonselective amylin receptors (AMYR) and calcitonin G protein-coupled receptor (CTR) agonist. Cagrilintide induces significant weight loss and reduces food intake. Cagrilintide has the potential for the research of obesity.
M28198 Vazegepant Vazegepant (Zavegepant) is a first-in-class CGRP receptor antagonist with potential for acute studies in migraine.
M25531 α-CGRP, human TFA α-CGRP, human TFA is a regulatory neuropeptide of 37 amino acids. α-CGRP, human TFA can be used as a potent vasodilator.
M22520 Galcanezumab Galcanezumab (LY 2951742) is a humanized IgG4 monoclonal antibody against the CGRP ligand.
M13935 Rat CGRP-(8-37) Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist.
M13933 MK-3207 MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3.
M13932 HCGRP-(8-37) HCGRP-(8-37) is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor.
M10894 Ubrogepant Ubrogepant (MK-1602) is a novel oral calcitonin gene-associated peptide receptor (CGRP) antagonist with the potential to be used in acute migraine studies.
M10801 Calcitonin (salmon) Calcitonin salmon is a calcium-regulating hormone that is a dual agonist of amylin and calcitonin receptors that stimulate bone production and inhibit bone resorption.
M10785 Atogepant Atogepant (MK-8031) is an orally active and selective calcitonin gene–related peptide receptor (CGRP) antagonist. Atogepant can be used for the research of migraine.
M10372 Vazegepant hydrochloride Vazegepant (BHV-3500) hydrochloride is a first-in-class, high affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM). Vazegepant hydrochloride may be useful in the effective treatment of lung inflammation associated with COVID-19.
M9165 Rimegepant Rimegepant, also known as BMS-927711, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 0.027 nM.
M6504 Olcegepant (BIBN-4096) Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide (CGRP) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.
M5240 BAR 501 impurity
M5223 BAR501 BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 μM.
M3618 MK-0974 MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively.
M2133 MK-3207 hydrochloride MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.

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