| Cat.No. | Name | Information |
|---|---|---|
| M2628 | Dexmedetomidine | Dexmedetomidine is a potent and highly selective α-2 adrenergic receptor agonist with sedative effects. |
| M3057 | Terbutaline Sulfate | Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM. |
| M3752 | Phentolamine Mesylate | Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED). |
| M2420 | Labetalol hydrochloride | Labetalol hydrochloride is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors. |
| M13893 | Labetalol | Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist. |
| M41768 | Moprolol | Moprolol ((±)-Moprolol) is an beta-adrenergic receptor blocker, which can be used for research in essential hypertension. |
| M41767 | Norfenefrine hydrochloride | Norfenefrine hydrochloride is an orally active, endogenously found α-adrenergic agonist and can be used for the research of female stress incontinence. |
| M41766 | Benzquinamide hydrochloride | Benzquinamide (P2647) is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively. |
| M41765 | Spiroxatrine | Spiroxatrine (R 5188) is a selective, dual antagonist of 5-HT1α and α2-adrenergic, with the Ki values of 3.94, 224000, 118.5 nM for 5-HT1α, 5-HT1β and 5-HT2, respectively. |
| M41764 | Abediterol | Abediterol (LAS100977) is an inhaled long-acting β2-adrenoceptor agonist (LABA) and can be used for the research of asthma and chronic obstructive pulmonary disease (COPD). |
| M41635 | Etilefrine hydrochloride | Etilefrine hydrochloride is an orally active α adrenergic agonist. |
| M40941 | Guanadrel | Guanadrel is an orally active, spiroketal postganglionic adrenergic inhibitor containing a spirocyclic moiety in its structure, which may be used in studies related to hypertension. |
| M40721 | Mabuterol | Mabuterol is a selective, orally active beta-2 adrenergic receptor (β2-AR) agonist. Mabuterol inhibits PDGF-BB-induced cell proliferation, increased intracellular Ca2+, and Drp-1, cyclinD1, and PCNA protein expression, and enhances Mfn-2 expression. Can be used in studies of airway obstruction and chronic obstructive pulmonary disease (COPD). |
| M38956 | Dicentrine | Dicentrine is a natural product isolated from the plant Stephania epigaea Lo with antihypertensive effect. Dicentrine is an α1-adrenoceptor antagonist which has effective against human hyperplastic prostates. |
| M38955 | Terbutaline | Terbutaline is an orally active β2-adrenergic receptor agonist and an active metabolite of bambuterol. Terbutaline can be used in asthma symptom research. |
| M38954 | Clenbuterol | Clenbuterol (NAB-365) is a β2-adrenergic receptor agonist with an EC50 of 31.9 nM. Clenbuterol is a very potent inhibitor of the lipopolysaccharide (LPS)-induced release of TNF-α and IL-1β. Clenbuterol can inhibit the inflammatory process. Clenbuterol is a bronchodilator. |
| M31211 | ST91 | ST91 is a α2-adrenoceptor (α2AR) agonist. ST91 activates both α2AAR and non-α2AAR subtypes to produce spinal antinociception. |
| M31210 | Ractopamine | Ractopamine is a potent β-adrenergic receptor (βAR) agonist with Kd value of ~25 nM for pig β1AR and β2AR. Ractopamine is linked to protein metabolism. |
| M31209 | Hydroxybupropion | Hydroxybupropion is the major active metabolite of Bupropion. Hydroxybupropion inhibits norepinephrine uptake with an IC50 value of 1.7 μM. Hydroxybupropion is also a nACh receptor antagonist. |
| M30990 | Adrenalone | Adrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic. Adrenalone is an inhibitor of dopamine β oxidase. Adrenalone is chemically similar to known norepinephrine transporter (NET) ligands with an IC50 of 36.9 μM. |
| M30933 | Levobetaxolol | Levobetaxolol is a potent and high affinity β-adrenergic antagonist with IC50 values of 33.2, 2970, 709 nM for guinea pig atrial β1, tracheal β2 and rat colonic β3 receptors, respectively. Levobetaxolol reduces IOP (intraocular pressure). Levobetaxolol exhibits a micromolar affinity for L-type Ca21-channels. Levobetaxolol decreases the effects of ischaemia/reperfusion injury in rats. Levobetaxolol has the potential for the research of glaucoma. |
| M30892 | Timolol hemihydrate | Timolol (hemihydrate) is a β-blocker available for both topical and systemic administration. Timolol (hemihydrate) is primarily used to reduce intraocular pressure with open-angle glaucoma and ocular hypertension and Timolol (hemihydrate) also has cardioprotective effect. |
| M30852 | Abanoquil | Abanoquil (U-K52046), an potent and selective α-1 adrenoceptor antagonist, is an anti-arrhythmic agent. Abanoquil can be used for erectile dysfunction research. |
| M30832 | ONO-2952 | ONO-2952 is a potent, selective and orally active translocator protein 18 kDa (TSPO) antagonist with Ki of 0.33-9.30 nM for rat and human TSPO. ONO-2952 is more selective for TSPO than other receptors, transporters, ion channels and enzymes. ONO-2952 exerts its anti-stress effects through inhibition of excessive activation of noradrenergic system in the brain without the amnesic effect. ONO-2952 has the potential for irritable bowel syndrome treatment. |
| M30722 | PF-610355 | PF-610355 is a long-acting inhaled β2-adrenoreceptor agonist, with an EC50 of 0.26 nM. PF-610355 has the potential for the study of asthma and COPD. |
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