| Cat.No. | Name | Information |
|---|---|---|
| M2628 | Dexmedetomidine | Dexmedetomidine is a potent and highly selective α-2 adrenergic receptor agonist with sedative effects. |
| M3057 | Terbutaline Sulfate | Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM. |
| M3752 | Phentolamine Mesylate | Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED). |
| M30333 | Bevantolol | Bevantolol is a selective β-1 adrenoceptor antagonist. Bevantolol can be used for the research of angina pectoris and hypertension. |
| M30286 | DL 071IT | DL 071IT is a potent non-selective beta-adrenergic receptor blocker. DL 071IT exhibits intrinsic sympathomimetic activity and weak membrane stabilizing activity. DL 071IT reduces exercise heart rate and systolic blood pressure, and even significantly lowers resting heart rate. |
| M30282 | Pronethalol | Pronethalol ((±)-Pronethalo) is a non-selective β-adrenergic antagonist. Pronethalol is a potent inhibitor of Sox2 expression. Pronethalol protects against and to reverse Digitalis-induced ventricular arrhythmias and limits the cerebral arteriovenous malformation (AVMs). |
| M30268 | Cimaterol | Cimaterol (CL 263780) is a β-adrenergic agonist on energy metabolism in ob/ob mice. The Kd for Cimaterol binding to the L6 β-receptor is 26 nM which is compatible with its EC50 for the stimulation of protein synthesis (approx 5 nM). |
| M30248 | TD-5471 hydrochloride | TD-5471 hydrochloride is a potent and selective full agonist of the human β2-adrenoceptor. |
| M30236 | Alloyohimbine | Alloyohimbine, an alkaloid, is a selective α2-adrenoceptor antagonist with K Dα1, K Dα2 of 0.28 μM and 0.006 μM, respectively. |
| M30220 | Naphazoline nitrate | Naphazoline (Naphthazoline) nitrate is an α-adrenergic receptor agonist. Naphazoline nitrate reduces vascular hyperpermeability and promotes vasoconstriction. Naphazoline nitrate reduces the levels of inflammatory factors (TNF-α, IL-1β and IL-6), cytokines (IFN-γ and IL-4), IgE, GMCSF, and NGF。Naphazoline nitrate can be used for non-bacterial conjunctivitis research. |
| M30212 | Pronethalol hydrochloride | Pronethalol ((±)-Pronethalo) is a non-selective β-adrenergic antagonist. Pronethalol is a potent inhibitor of Sox2 expression. Pronethalol protects against and to reverse Digitalis-induced ventricular arrhythmias, and limits the cerebral arteriovenous malformation (AVMs). |
| M30198 | Mezilamine | Mezilamine is a potent antidopaminergic agent. Mezilamine induces a concentration dependent increase in the electrically stimulated overflow of 3H-noradrenaline from rat cortical slices, without affecting the basal overflow. Mezilamine acts as a presynaptic α-adrenoceptor antagonist and a postsynaptic α-adrenoceptor agonist. |
| M30002 | Zinterol | Zinterol (MJ 9184) is a potent and selective β2-adrenoceptor agonist. Zinterol increases ICa in a concentration-dependent manner with an EC50 of 2.2 nM. |
| M29947 | Levalbuterol | Levalbuterol ((R)-Albuterol; (R)-Salbutamol) is a short-acting β2-adrenergic receptor agonist and the active (R)-enantiomer of Salbutamol. Levalbuterol is a more potent bronchodilator than Salbutamol and has the potential for the treatment of COPD. |
| M29347 | N-5984 | N-5984 (KRP-204) is a potent and selective agonist of β3-adrenergic receptor. N-5984 has the potential for developing as one of the clinically effective drugs for obesity and diabetes mellitus. |
| M29250 | L-796568 | L-796568 is a β(3)-adrenergic receptor agonist. L-796568 can be used for the research of obesity. |
| M28518 | Carmoterol | Carmoterol is a highly potent, selective and long-acting β2-adrenoceptor agonist with the pEC50 of 10.19. Carmoterol has 53 times higher affinity for the β2-adrenoceptors than for the β1-adrenoceptors. Carmoterol can be used for the research of asthma and chronic obstructive pulmonary disease (COPD). |
| M28475 | Piribedil dihydrochloride | Piribedil dihydrochloride is a potent and orally active dopamine D2 and dopamine D3 agonist. Piribedil dihydrochloride is also a α2-adrenoceptors antagonist. Piribedil dihydrochloride can inhibit MLL1 methyltransferase activity (EC50: 0.18 μM). Piribedil dihydrochloride has the potential for the research of parkinson's disease, circulatory disorders, cancers. |
| M28242 | Piperoxan hydrochloride | Piperoxan (Benodaine) hydrochloride is an α2 adrenoceptor antagonist. Piperoxan hydrochloride is the first-generation antihistamine. |
| M28053 | Arformoterol maleate | Arformoterol ((R,R)-Formoterol) maleate, the (R,R)-enantiomer of Formoterol, is a long-acting β2-adrenergic receptor (β2-AR) agonist, with a Kd of 2.9 nM. Arformoterol maleate can be used for the research of chronic obstructive pulmonary disease (COPD). |
| M27928 | BI-167107 | BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM. |
| M27734 | Butyryltimolol | Butyryltimolol is the active precursor compound of Timolol, and is also a β-adrenergic (β-AR) blocker, which can pass through the cornea of the eye, and is enzymatically hydrolyzed to produce Timolol after entering the eye. |
| M25455 | Butoxamine hydrochloride | Butoxamine hydrochloride is a specific β2-adrenergic receptor blocker. |
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2023 AbMole BioScience. All Rights Reserved.
