Inhibitors
Cat.No. | Name | Information |
---|---|---|
M9329 | Fenoterol | Fenoterol is a β2 adrenoreceptor agonist with bronchodilator activity. |
M9264 | Norepinephrine | Norepinephrine is generally considered to be a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM. |
M9201 | Vibegron | Vibegron is a potent and selective beta 3 adrenergic receptor agonist. |
M7848 | ICI 118,551 hydrochloride | ICI 118,551 hydrochloride is a highly selective β2-adrenoceptor antagonist. |
M7743 | Dobutamine hydrochloride | Dobutamine hydrochloride is a selective β1-AR agonist. |
M6887 | L-755,507 | L-755,507 is a very potent and selective β3 partial agonist. |
M6291 | 5-Iodotubercidin | 5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinase, phosphorylase kinase, PKA, CK2 and PKC. |
M6061 | Xylometazoline HCl | Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM. |
M6060 | Xylazine HCl | Xylazine is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant. |
M6019 | Tizanidine HCl | Tizanidine hydrochloride is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons. |
M6000 | Terazosin HCl | Terazosin is a selective alpha-1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). It works by blocking the action of adrenaline on smooth muscle of the bladder and the blood vessel walls. |
M5999 | Terazosin HCl Dihydrate | Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH). |
M5998 | Terazosin | Terazosin is a selective alpha1-antagonist used for treatment of symptoms of benign prostatic hyperplasia (BPH). |
M5988 | Tamsulosin | Tamsulosin is a selective α1 receptor antagonist. |
M5953 | Scopine HCl | Scopine Hcl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock. |
M5947 | Salmeterol Xinafoate | Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms. |
M5936 | Ritodrine HCl | Ritodrine HCl is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist. |
M5895 | Prazosin HCl | Prazosin HCl is a competitive alpha-1 adrenoceptor antagonist, used to treat high blood pressure or benign prostatic hyperplasia. |
M5894 | Prazosin | Prazosin is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder. |
M5822 | Noradrenaline bitartrate monohydrate | Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator. |
M5808 | Naphazoline HCl | Naphazoline HCl is an ocular vasoconstrictor and imidazoline derivative sympathomimetic amine. |
M5785 | Metoprolol Tartrate | Metoprolol Tartrate is a selective β1 receptor blocker medication, used to treat hypertension and heart failure. |
M5784 | Metoprolol Succinate | Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension. |
M5781 | Methoxyphenamine HCl | Methoxyphenamine Hydrochloride is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator. |
M5720 | Ivabradine HCl | Ivabradine HCl, a new If inhibitor with IC 50 of 2.9 μM which acts specifically on the pacemaker activity of the sinoatrial node, is a pure heart rate lowering agent. |
M5685 | Guanfacine HCl | Guanfacine Hcl, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over α2B-adrenoceptors. |
M5644 | Fenoterol hydrobromide | Fenoterol hydrobromide is a β 2 adrenergic agonist designed to open up the airways to the lungs, is classed as sympathomimetic β2 agonist and asthma medication. |
M5616 | Epinephrine bitartrate | Epinephrine bitartrate is an alpha- and beta-adrenergic receptor stimulator. |
M5593 | Doxazosin Mesylate | Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia. |
M5471 | Buflomedil HCl | Buflomedil HCl is a vasodilator used to treat claudication or the symptoms of peripheral arterial disease; A nonselective alpha adrenergic receptor inhibitor |
M5462 | Bisoprolol fumarate | Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker. |
M5459 | Atipamezole HCl | Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride is hydrochloride form of atipamezole. |
M5456 | B-HT 920 | B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity. |
M5453 | Betaxolol | Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma. |
M5429 | Atipamezole | Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. |
M5428 | Atenolol | Atenolol is a selective β1 receptor antagonist. |
M5405 | Amezinium methylsulfate | Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition ofnoradrenaline and tyramine uptake. |
M5239 | GSK-961081 | GSK961081 is a novel inhaled bifunctional compound that was designed to exhibit dual muscarinic antagonist and β2-adrenoceptor agonist (MABA) pharmacology with the potential to deliver optimal bronchodilation after inhalation dosing via two validated mechanisms in one molecule. |
M5116 | Formoterol Hemifumarate | Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease. |
M4821 | Vilanterol trifenatate | Vilanterol trifenatate is a novel, long-acting β(2)-adrenoceptor (β(2)-AR) agonist with 24 h activity. |
M4820 | Vilanterol | Vilanterol is a novel, inhaled, long-acting β(2) agonist with inherent 24-h activity under development as a once-daily combination therapy with an inhaled corticosteroid for COPD and asthma. |
M4593 | Yohimbine-Hydrochloride | Yohimbine hydrochloride is an α2-adrenergic receptor antagonist. |
M3752 | Phentolamine Mesylate | Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED). |
M3662 | Bambuterol hydrochloride | Bambuterol hydrochloride is a potent β-adrenoceptor agonist, used in the treatment of asthma. |
M3656 | Carteolol hydrochloride | Carteolol hydrochloride is a non-selective beta blocker which is used to treat glaucoma. |
M3605 | Salbutamol Sulfate | Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM. |
M3551 | Silodosin | Silodosin is an α1-adrenoceptor antagonist with high uroselectivity. |
M3509 | Nebivolol | Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM. |
M3482 | Carvedilol | Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation. |
M3457 | Naftopidil | Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM. |
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