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Abmole Inhibitor Catalog 2017

Adrenergic Receptor Adrenergic Receptor

Inhibitors

Cat.No.  Name Information
M6061 Xylometazoline HCl Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM.
M6060 Xylazine HCl Xylazine is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant.
M6019 Tizanidine HCl Tizanidine hydrochloride is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
M6000 Terazosin HCl Terazosin is a selective alpha-1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). It works by blocking the action of adrenaline on smooth muscle of the bladder and the blood vessel walls.
M5999 Terazosin HCl Dihydrate Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
M5998 Terazosin Terazosin is a selective alpha1-antagonist used for treatment of symptoms of benign prostatic hyperplasia (BPH).
M5988 Tamsulosin Tamsulosin is a selective α1 receptor antagonist.
M5953 Scopine HCl Scopine Hcl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
M5947 Salmeterol Xinafoate Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms.
M5936 Ritodrine HCl Ritodrine HCl is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist.
M5895 Prazosin HCl Prazosin HCl is a competitive alpha-1 adrenoceptor antagonist, used to treat high blood pressure or benign prostatic hyperplasia.
M5894 Prazosin Prazosin is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder.
M5822 Noradrenaline bitartrate monohydrate Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.
M5808 Naphazoline HCl Naphazoline HCl is an ocular vasoconstrictor and imidazoline derivative sympathomimetic amine.
M5785 Metoprolol Tartrate Metoprolol Tartrate is a selective β1 receptor blocker medication, used to treat hypertension and heart failure.
M5784 Metoprolol Succinate Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension.
M5781 Methoxyphenamine HCl Methoxyphenamine Hydrochloride is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
M5726 L-Adrenaline L-Adrenaline belongs to a group of the compounds known as catecholamines.
M5720 Ivabradine HCl Ivabradine HCl, a new If inhibitor with IC 50 of 2.9 μM which acts specifically on the pacemaker activity of the sinoatrial node, is a pure heart rate lowering agent.
M5685 Guanfacine HCl Guanfacine Hcl, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over α2B-adrenoceptors.
M5644 Fenoterol Fenoterol hydrobromide is a β 2 adrenergic agonist designed to open up the airways to the lungs, is classed as sympathomimetic β2 agonist and asthma medication.
M5616 Epinephrine bitartrate Epinephrine bitartrate is an alpha- and beta-adrenergic receptor stimulator.
M5593 Doxazosin Mesylate Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia.
M5471 Buflomedil HCl Buflomedil HCl is a vasodilator used to treat claudication or the symptoms of peripheral arterial disease; A nonselective alpha adrenergic receptor inhibitor
M5462 Bisoprolol fumarate Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker.
M5459 Atipamezole HCl Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride is hydrochloride form of atipamezole.
M5456 B-HT 920 B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity.
M5453 Betaxolol Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
M5429 Atipamezole Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
M5428 Atenolol Atenolol is a selective β1 receptor antagonist.
M5405 Amezinium methylsulfate Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition ofnoradrenaline and tyramine uptake.
M5239 GSK-961081 GSK961081 is a novel inhaled bifunctional compound that was designed to exhibit dual muscarinic antagonist and β2-adrenoceptor agonist (MABA) pharmacology with the potential to deliver optimal bronchodilation after inhalation dosing via two validated mechanisms in one molecule.
M5116 Formoterol Hemifumarate Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease.
M4821 Vilanterol trifenatate Vilanterol trifenatate is a novel, long-acting β(2)-adrenoceptor (β(2)-AR) agonist with 24 h activity.
M4820 Vilanterol Vilanterol is a novel, inhaled, long-acting β(2) agonist with inherent 24-h activity under development as a once-daily combination therapy with an inhaled corticosteroid for COPD and asthma.
M3752 Phentolamine Mesylate Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED).
M3662 Bambuterol hydrochloride Bambuterol hydrochloride is a potent β-adrenoceptor agonist, used in the treatment of asthma.
M3656 Carteolol hydrochloride Carteolol hydrochloride is a non-selective beta blocker which is used to treat glaucoma.
M3605 Salbutamol Sulfate Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.
M3551 Silodosin Silodosin is an α1-adrenoceptor antagonist with high uroselectivity.
M3509 Nebivolol Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.
M3482 Carvedilol Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.
M3457 Naftopidil Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
M3413 Phenoxybenzamine hydrochloride Phenoxybenzamine hydrochloride is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM.
M3411 Sotalol Sotalol is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM.
M3408 Maprotiline hydrochloride Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.
M3372 Clonidine hydrochloride Clonidine hydrochloride is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg.
M3370 Oxymetazoline hydrochloride Oxymetazoline hydrochloride is an α1 and α2 adrenergic receptor agonist.
M3330 Phenylephrine hydrochloride Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist.
M3186 Isoprenaline hydrochloride Isoproterenol hydrochloride is a non-selective β-adrenoceptor, inhibits the 3H-inositol phosphate accumulation with IC50 of 0.08 μM.


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