Catalog

Adrenergic Receptor Adrenergic Receptor

Inhibitors

Cat.No.	Name	Information
M9264	Norepinephrine	Norepinephrine is generally considered to be a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM.
M9201	Vibegron	Vibegron is a potent and selective beta 3 adrenergic receptor agonist.
M6887	L-755,507	L-755,507 is a very potent and selective β ₃ partial agonist.
M6291	5-Iodotubercidin	5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinase, phosphorylase kinase, PKA, CK2 and PKC.
M6061	Xylometazoline HCl	Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM.
M6060	Xylazine HCl	Xylazine is an α2-Adrenergic receptor agonist, used as a sedative and muscle relaxant.
M6019	Tizanidine HCl	Tizanidine hydrochloride is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
M6000	Terazosin HCl	Terazosin is a selective alpha-1 antagonist used for treatment of symptoms of an enlarged prostate (BPH). It works by blocking the action of adrenaline on smooth muscle of the bladder and the blood vessel walls.
M5999	Terazosin HCl Dihydrate	Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
M5998	Terazosin	Terazosin is a selective alpha1-antagonist used for treatment of symptoms of benign prostatic hyperplasia (BPH).
M5988	Tamsulosin	Tamsulosin is a selective α1 receptor antagonist.
M5953	Scopine HCl	Scopine Hcl salt is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
M5947	Salmeterol Xinafoate	Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms.
M5936	Ritodrine HCl	Ritodrine HCl is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist.
M5895	Prazosin HCl	Prazosin HCl is a competitive alpha-1 adrenoceptor antagonist, used to treat high blood pressure or benign prostatic hyperplasia.
M5894	Prazosin	Prazosin is an alpha-adrenergic blocker and is a sympatholytic drug used to treat high blood pressure and anxiety, PTSD, and panic disorder.
M5822	Noradrenaline bitartrate monohydrate	Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.
M5808	Naphazoline HCl	Naphazoline HCl is an ocular vasoconstrictor and imidazoline derivative sympathomimetic amine.
M5785	Metoprolol Tartrate	Metoprolol Tartrate is a selective β1 receptor blocker medication, used to treat hypertension and heart failure.
M5784	Metoprolol Succinate	Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension.
M5781	Methoxyphenamine HCl	Methoxyphenamine Hydrochloride is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
M5720	Ivabradine HCl	Ivabradine HCl, a new If inhibitor with IC 50 of 2.9 μM which acts specifically on the pacemaker activity of the sinoatrial node, is a pure heart rate lowering agent.
M5685	Guanfacine HCl	Guanfacine Hcl, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over α2B-adrenoceptors.
M5644	Fenoterol hydrobromide	Fenoterol hydrobromide is a β 2 adrenergic agonist designed to open up the airways to the lungs, is classed as sympathomimetic β2 agonist and asthma medication.
M5616	Epinephrine bitartrate	Epinephrine bitartrate is an alpha- and beta-adrenergic receptor stimulator.
M5593	Doxazosin Mesylate	Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia.
M5471	Buflomedil HCl	Buflomedil HCl is a vasodilator used to treat claudication or the symptoms of peripheral arterial disease; A nonselective alpha adrenergic receptor inhibitor
M5462	Bisoprolol fumarate	Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker.
M5459	Atipamezole HCl	Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride is hydrochloride form of atipamezole.
M5456	B-HT 920	B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity.
M5453	Betaxolol	Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
M5429	Atipamezole	Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
M5428	Atenolol	Atenolol is a selective β1 receptor antagonist.
M5405	Amezinium methylsulfate	Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition ofnoradrenaline and tyramine uptake.
M5239	GSK-961081	GSK961081 is a novel inhaled bifunctional compound that was designed to exhibit dual muscarinic antagonist and β2-adrenoceptor agonist (MABA) pharmacology with the potential to deliver optimal bronchodilation after inhalation dosing via two validated mechanisms in one molecule.
M5116	Formoterol Hemifumarate	Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease.
M4821	Vilanterol trifenatate	Vilanterol trifenatate is a novel, long-acting β(2)-adrenoceptor (β(2)-AR) agonist with 24 h activity.
M4820	Vilanterol	Vilanterol is a novel, inhaled, long-acting β(2) agonist with inherent 24-h activity under development as a once-daily combination therapy with an inhaled corticosteroid for COPD and asthma.
M3752	Phentolamine Mesylate	Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED).
M3662	Bambuterol hydrochloride	Bambuterol hydrochloride is a potent β-adrenoceptor agonist, used in the treatment of asthma.
M3656	Carteolol hydrochloride	Carteolol hydrochloride is a non-selective beta blocker which is used to treat glaucoma.
M3605	Salbutamol Sulfate	Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.
M3551	Silodosin	Silodosin is an α1-adrenoceptor antagonist with high uroselectivity.
M3509	Nebivolol	Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.
M3482	Carvedilol	Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.
M3457	Naftopidil	Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
M3413	Phenoxybenzamine hydrochloride	Phenoxybenzamine hydrochloride is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM.
M3411	Sotalol	Sotalol is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM.
M3408	Maprotiline hydrochloride	Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.
M3372	Clonidine hydrochloride	Clonidine hydrochloride is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg.

Signaling Pathways

Product Type

Adrenergic Receptor Adrenergic Receptor

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