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Abmole Inhibitor Catalog 2017

Adrenergic Receptor Adrenergic Receptor

Inhibitors

Cat.No.  Name Information
M5616 Epinephrine bitartrate Epinephrine bitartrate is an alpha- and beta-adrenergic receptor stimulator.
M5593 Doxazosin Mesylate Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia.
M5471 Buflomedil HCl Buflomedil HCl is a vasodilator used to treat claudication or the symptoms of peripheral arterial disease; A nonselective alpha adrenergic receptor inhibitor
M5462 Bisoprolol fumarate Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker.
M5459 Atipamezole HCl Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride is hydrochloride form of atipamezole.
M5456 B-HT 920 B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity.
M5453 Betaxolol Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
M5429 Atipamezole Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
M5428 Atenolol Atenolol is a selective β1 receptor antagonist.
M5405 Amezinium methylsulfate Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition ofnoradrenaline and tyramine uptake.
M5239 GSK-961081 GSK961081 is a novel inhaled bifunctional compound that was designed to exhibit dual muscarinic antagonist and β2-adrenoceptor agonist (MABA) pharmacology with the potential to deliver optimal bronchodilation after inhalation dosing via two validated mechanisms in one molecule.
M5116 Formoterol Hemifumarate Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease.
M4821 Vilanterol trifenatate Vilanterol trifenatate is a novel, long-acting β(2)-adrenoceptor (β(2)-AR) agonist with 24 h activity.
M4820 Vilanterol Vilanterol is a novel, inhaled, long-acting β(2) agonist with inherent 24-h activity under development as a once-daily combination therapy with an inhaled corticosteroid for COPD and asthma.
M3752 Phentolamine Mesylate Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED).
M3662 Bambuterol hydrochloride Bambuterol hydrochloride is a potent β-adrenoceptor agonist, used in the treatment of asthma.
M3656 Carteolol hydrochloride Carteolol hydrochloride is a non-selective beta blocker which is used to treat glaucoma.
M3605 Salbutamol Sulfate Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.
M3551 Silodosin Silodosin is an α1-adrenoceptor antagonist with high uroselectivity.
M3509 Nebivolol Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.
M3482 Carvedilol Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.
M3457 Naftopidil Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
M3413 Phenoxybenzamine hydrochloride Phenoxybenzamine hydrochloride is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM.
M3411 Sotalol Sotalol is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM.
M3408 Maprotiline hydrochloride Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.
M3372 Clonidine hydrochloride Clonidine hydrochloride is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg.
M3370 Oxymetazoline hydrochloride Oxymetazoline hydrochloride is an α1 and α2 adrenergic receptor agonist.
M3330 Phenylephrine hydrochloride Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist.
M3186 Isoprenaline hydrochloride Isoproterenol hydrochloride is a non-selective β-adrenoceptor, inhibits the 3H-inositol phosphate accumulation with IC50 of 0.08 μM.
M3076 Tolazoline hydrochloride Tolazoline is a non-selective competitive α-adrenergic receptor antagonist.
M3072 Timolol Maleate Timolol Maleate is a non-selective, beta-adrenergic receptor antagonist for β1/β2 with Ki of 1.97 nM/2.0 nM.
M3060 Tetrahydrozoline hydrochloride Tetrahydrozoline hydrochloride is an imidazoline derivative with alpha receptor agonist activity.
M3057 Terbutaline Sulfate Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM.
M3043 Synephrine hydrochloride SynephrineHCl (Oxedrine, p-Synephrine) is a sympathomimetic α-adrenergic receptor (AR) agonist.
M2964 Propranolol hydrochloride Propranolol hydrochloride is a competitive non-selective beta-adrenergic receptors inhibitor with IC50 of 12 nM.
M2834 Medetomidine hydrochloride Medetomidine is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
M2808 Levalbuterol hydrochloride Levalbuterol hydrochloride is a relatively selective beta2-adrenergic receptor agonist used for the treatment of asthma.
M2772 Indacaterol Maleate Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.
M2738 Guanabenz Acetate Guanabenz Acetate is an selective agonist of α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor with pEC50 of 8.25, 7.01 and ~5, respectively.
M2672 Epinephrine hydrochloride Epinephrine hydrochloride is a hormone and a neurotransmitter.
M2628 Dexmedetomidine Dexmedetomidine is a sedative medication used by intensive care units and anesthetists.
M2468 Brimonidine Tartrate Brimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.
M2420 Labetalol hydrochloride Labetalol hydrochloride is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors.
M2370 Adrenalone hydrochloride Adrenalone is an adrenergic agonist used as a topical vasoconstrictor and hemostatic, mainly acts on alpha-1 adrenergic receptors.
M2365 Acebutolol hydrochloride Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.
M2077 Detomidine hydrochloride Detomidine hydrochloride is a nonnarcotic, synthetic alpha-2 adrenoreceptor agonist.
M2069 Mirabegron Mirabegron (YM178) is a potent and selective β(3)-adrenoceptor agonist with EC50 of 22.4 nM.
M1889 Tamsulosin hydrochloride Tamsulosin is a new, highly selective α1A-adrenoceptor antagonist.

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