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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M13902 | Yohimbine | Yohimbine is a potent and relatively nonselective alpha 2-adrenergic receptor (AR) antagonist, with IC50 of 0.6 μM. |
| M13901 | Tulobuterol hydrochloride | Tulobuterol hydrochloride (C-78) is a long-acting β2-adrenoceptor agonist, which reduces the frequency of exacerbations of chronic obstructive pulmonary disease and bronchial asthma. |
| M13900 | Tulobuterol | Tulobuterol (C-78 free base) is a long-acting β2-adrenoceptor agonist, which reduces the frequency of exacerbations of chronic obstructive pulmonary disease and bronchial asthma. |
| M13899 | SR59230A hydrochloride | SR59230A hydrochloride is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50s of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively. |
| M13898 | Penbutolol sulfate | Penbutolol sulfate is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making it a non-selective β blocker. Penbutolol is a sympathomimetic drug，used in the treatment of high blood pressure. |
| M13897 | Olodaterol hydrochloride | Olodaterol (BI1744) hydrochloride is a selective, long acting β2-adrenoceptor (β2-AR) agonist (EC50=0.1 nM and pKi= 9.14 for human β2-adrenoceptor, respectively). |
| M13896 | Norepinephrine hydrochloride | Norepinephrine (Levarterenol; L-Noradrenaline) hydrochloride is a potent adrenergic receptor (AR) agonist. Norepinephrine activates α1, α2, β1 receptors. |
| M13895 | Metipranolol hydrochloride | Metipranolol hydrochloride is a non-selective β adrenergic receptor blocking agent. |
| M13894 | L-Epinephrine | L-Epinephrine is a hormone secreted by the medulla of the adrenal glands. L-Epinephrine is an α-adrenergic and β-adrenergic receptor agonist. |
| M13893 | Labetalol | Labetalol (AH5158) is an orally active selective α1- and non-selective β-adrenergic receptors competitive antagonist. |
| M13892 | Methyldopa hydrate | Methyldopa hydrate (L-(-)-α-Methyldopa hydrate), a potent antihyoertensive agent, is an alpha-adrenergic agonist (selective for α2-adrenergic receptors). |
| M13891 | Arformoterol | Arformoterol ((R,R)-Formoterol), the (R,R)-enantiomer of Formoterol, is a long-acting β2-adrenergic receptor (β2-AR) agonist, with a Kd of 2.9 nM. |
| M13890 | Clonidine | Clonidine is an alpha 2-adrenergic agonist. |
| M13889 | CL 316243 | CL316243 is a highly potent selective β3-adrenoceptor agonist with a EC50 of 3 nM, but is an extremely poor to β1/2- receptors.CL316243 is a effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate. |
| M13888 | Bufuralol hydrochloride | Bufuralol hydrochloride (Ro 3-4787 hydrochloride) is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate. |
| M11540 | Propranolol | Propranolol is a non-selective β-adrenergic receptor (βAR) antagonist, which has high affinity for β1AR and β2AR with Ki value of 1.8 nM and 0.8 nM, respectively. Propranolol inhibited the binding of [3H]-DHA to rat meninges with an IC50 of 12 nM. |
| M11289 | Solabegron | Solabegron (GW 427353) is a selective agonist of β3 adrenergic receptor (β3-AR). The EC50 value of Solabegron was 22 nM in Chinese hamster ovarian cells. It can be used to study overactive bladder and irritable bowel syndrome. |
| M10994 | Higenamine hydrochloride | Higenamine hydrochloride (Norcoclaurine hydrochloride) is a beta2-AR agonist that is a key ingredient in the Aconitum of Chinese medicine used in heart failure-related studies. Higenamine hydrochloride (Norcoclaurine hydrochloride) has an anti-apoptotic effect. |
| M10684 | Phenylephrine | (R)-(-)-Phenylephrine is a selective α1- adrenergic receptor agonists, mainly used as decongestants. |
| M10654 | Ajmalicine (Raubasine) | Ajmalicine (Raubasine) is an adrenolytic agent which preferentially blocks alpha 1-adrenoceptor than alpha 2-adrenoceptor. Ajmalicine (Raubasine) is an reversible non-competitive nicotine receptor antagonist with an IC50 of 72.3 μM. |
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