Free shipping on all orders over $ 500

Adrenergic Receptor Adrenergic Receptor

Inhibitors

Cat.No.  Name Information
M2628 Dexmedetomidine Dexmedetomidine is a potent and highly selective α-2 adrenergic receptor agonist with sedative effects.
M5239 GSK-961081 GSK961081 is a novel inhaled bifunctional compound that was designed to exhibit dual muscarinic antagonist and β2-adrenoceptor agonist (MABA) pharmacology with the potential to deliver optimal bronchodilation after inhalation dosing via two validated mechanisms in one molecule.
M5116 Formoterol Hemifumarate Formoterol Hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist used in the management of asthma and chronic obstructive pulmonary disease.
M4821 Vilanterol trifenatate Vilanterol trifenatate is a novel, long-acting β(2)-adrenoceptor (β(2)-AR) agonist with 24 h activity.
M4820 Vilanterol Vilanterol(GW642444, Veranterol) is a long-acting β2-AR agonist. PEC50 of β2-AR, β1-AR and β3-AR were 10.37, 6.98, 7.36, respectively.
M4593 Yohimbine-Hydrochloride Yohimbine hydrochloride is an α2-adrenergic receptor antagonist.
M4447 3-Hydroxy-4-methoxycinnamic-acid Isoferulic acid (3-Hydroxy-4-methoxycinnamic acid) is a kind of cinnamic acid derivative with anti - diabetes activity. Isoferulic acid (3-hydroxy-4-methoxycinnamic acid) binds and activates α 1-adrenergic receptor (IC50=1.4 μM), Enhanced β -endorphin secretion (EC50=52.2 nM) and increased in vitro glucose use. Isoferulic acid also has activity against influenza virus.
M3752 Phentolamine Mesylate Phentolamine mesylate is an orally active, rapid-acting alpha-adrenergic receptor antagonist, for the treatment of men suffering from erectile dysfunction (ED).
M3662 Bambuterol hydrochloride Bambuterol hydrochloride is an effective β -adrenergic receptor agonist.
M3656 Carteolol hydrochloride Carteolol hydrochloride is a non-selective β -blocker used to study glaucoma.
M3605 Salbutamol Sulfate Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.
M3551 Silodosin Silodosin is an α1-adrenoceptor antagonist with high uroselectivity.
M3509 Nebivolol Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.
M3482 Carvedilol Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.
M3457 Naftopidil Naftopidil is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
M3413 Phenoxybenzamine hydrochloride Phenoxybenzamine hydrochloride is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM.
M3411 Sotalol Sotalol is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM.
M3408 Maprotiline hydrochloride Maprotiline hydrochloride is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.
M3372 Clonidine hydrochloride Clonidine hydrochloride is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg.
M3370 Oxymetazoline hydrochloride Oxymetazoline hydrochloride is an α1 and α2 adrenergic receptor agonist.
M3330 Phenylephrine hydrochloride Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist.



Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2020 AbMole BioScience. All Rights Reserved.