TS-011 - Search Results | AbMole BioScience

About 6 results found for searched term "TS-011" (0.127 seconds)

Cat.No.	Name	Target
M2201	TSR-011	ALK
	Belizatinib
	TSR-011 is a potent, orally available ALK inhibitor.
M45354	TS-011	Cytochrome P450 (e.g. CYP17)
	TS-011 is a selective inhibitor of 20-hydroxyeicosatetraenoic acid (20-HETE) synthesis.
M5854	SB 277011 Hydrochloride	Dopamine Receptor
	Ligands acting as DRD3 antagonists (SB 277011-A) has shown some promise for reducing the influence of drug-associated cues on motivational behaviour.
M30420	3M-011	TLR
	3M-011 is a potent dual toll-like receptor TLR7/8 agonist and a cytokine inducer. 3M-011 significantly inhibits H3N2 influenza viral replication in the nasal cavity. 3M-011 is also a potent adjuvant to radiotherapy that induces local and profound systemic immune responses during radiotherapy. 3M-011 strongly has antitumor action.
M45398	MSU-42011	RAR/RXR
	MSU-42011 is an orally active retinoid X receptor-like (RXR) agonist that potently inhibits the expression of iNOS as well as p-ERK protein levels. In addition, MSU-42011 has immunomodulatory and antitumor activities for cancer research.
M57237	AZ12601011	TGF-β Receptor
	AZ12601011 is an orally active, selective TGFBR1 kinase inhibitor with an IC50 of 18 nM and a Kd of 2.9 nM. AZ12601011 inhibits phosphorylation of SMAD2 via selectively inhibiting ALK4, TGFBR1, and ALK7. AZ12601011 inhibits mammary tumor growth.