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 About 24 results found for searched term "PI3K" (0.051 seconds)

Cat.No.  Name Target
M5343 Voxtalisib Analogue PI3K
PI3K-IN-1; XL-147 derivative 1; SAR245409
PI3K-IN-1 (XL-147 derivative 1) is a dual inhibitor of mTOR/PI3K, mostly for p110γ with IC50 of 9 nM; also inhibits DNA-PK and mTOR. Phase 1/2.
M10443 Linperlisib (YY-20394) PI3K
YY-20394; PI3Kδ-IN-2
Linperlisib, also known as YY-20394 and PI3Kδ-IN-2, is a potent and selective PI3Kδ inhibitor.
M14854 PI3K/mTOR Inhibitor-2 PI3K
PI3K/mTOR Inhibitor-2 is a potent dual pan-PI3K/mTOR inhibitor with IC50s of 3.4/34/16/1 nM for PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ and 4.7 nM for mTOR. Antitumor activity.
M20632 Selective PI3Kδ Inhibitor 1 (compound 7n) PI3K
Selective PI3Kδ Inhibitor 1 (compound 7n) is an inhibitor of PI3Kδ with an IC50 of 0.9 nM and >1000-fold selectivity against other class I PI3K isoforms [PI3K α/γ/β=3670/1460/21300 nM].
M28008 BEBT-908 PI3K
PI3Kα inhibitor 1
BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor with an IC50<0.1 μM, it also inhibits HDAC (0.1 μM≤IC50≤1 μM) .
M29360 PI3K-IN-10  PI3K
PI3K-IN-10 is a potent pan-PI3K inhibitor as a benzimidazole derivative.
M30007 PI3K-IN-32  PI3K
PI3K-IN-32 (compound 35) is a potent PI3K p110α inhibitor with an pIC50 of 6.85.
M43372 PI3K-IN-48 Akt
PI3K-IN-48 is a PI3K inhibitor with IC50 value of 1.55 ± 0.18 μM for A549 cells.
M43377 PI3Kδ-IN-16 Apoptosis
PI3Kδ-IN-16 is a potent and selective inhibitor of PI3Kδ.
M43388 PI3Kγ inhibitor 7 PI3K
PI3Kγ inhibitor 7 is a potent and orally active PI3Kγ inhibitor with IC50 values of 4768, 878.1, 3.42, 355.2 nM for PI3Kα, PI3Kβ, PI3Kγ, PI3Kδ, respectively.
M43390 IHMT-PI3K-455 PI3K
IHMT-PI3K-455 is a potent, selective, orally active PI3Kγ/δ dual inhibitor with IC50s of 7.1 nM and 0.57 nM for PI3Kγ and PI3Kδ, respectively.
M43391 PI3K-IN-47 PI3K
PI3K-IN-47 is a bivalent PI3K inhibitor (IC50: 0.44 nM for PI3Kα, 7.18 nM, 13.92 nM, 22.83 nM for PI3Kβ, PI3Kγ, PI3Kδ).
M43392 PI3K-IN-41 PI3K
PI3K-IN-41 is a photocaged compound, as well as a photocaged PI3K inhibitor (IC50=18.92 nM) with anticancer properties.
M43393 PI3Kδ-IN-12 PI3K
PI3Kδ-IN-12 is a PI3Kδ inhibitor (pIC50 = 5.8), with pKi values of 8.0/6.5/6.4/6.7 for PI3Kδ/γ/β/α, respectively.
M43398 PI3Kδ-IN-14 PI3K
PI3Kδ-IN-14 is a selective PI3Kδ inhibitor (IC50: 0.8 nM, Kd: 84.8 nM).
M43401 PI3Kα-IN-13 PI3K
PI3Kα-IN-13 is a PI3Kα inhibitor (IC50: 2.5 nM).
M43402 PI3Kδ-IN-13 PI3K
PI3Kδ-IN-13 is a PI3Kδ inhibitor (IC50=2.6 nM).
M55555 PI3K/Akt/CREB activator 1 PI3K
compound AE-18
PI3K/Akt/CREB activator 1 (compound AE-18) is a potent, orally active PI3K/Akt/CREB activator. PI3K/Akt/CREB activator 1 promotes neuronal proliferation, induced differentiation of Neuro-2a cells into a neuron-like morphology, and accelerated the establishment of axon-dendrite polarization of primary hippocampal neurons through upregulating brain-derived neurotrophic factor via the PI3K/Akt/CREB pathway.
M57083 PI3Kγ inhibitor AZ2  PI3K
PI3Kγ inhibitor AZ2 is a highly selective PI3Kγ inhibitor (The pIC50 value for PI3Kγ is 9.3).
M57078 PI3Kα-IN-22  PI3K
PI3Kα-IN-22 is an orally active, potent and selective inhibitor of PI3KαH1047R, with an IC50 of 1 nM for pAKT T47D AlphaLISA.
M57077 PI3K/AKT-IN-1  PI3K
PI3K/AKT-IN-1 is an effective PI3K/AKT dual inhibitor (IC50 of 6.99, 4.01 and 3.36 μM for PI3Kγ, PI3Kδ and AKT, respectively).
M57076 CHMFL-PI3KD-317  PI3K
CHMFL-PI3KD-317 is a highly potent, selective and orally active PI3Kδ inhibitor, with an IC50 of 6 nM, and exhibits over 10-1500 fold selectivity over other class I, II and III PIKK family isoforms.
M57075 PI3Kδ-IN-1  PI3K
PI3Kδ-IN-1 is a potent, selective, and efficacious PI3Kδ inhibitor with an IC50 of 1.7 nM.
M57074 PI3K/Akt/mTOR-IN-2  PI3K
PI3K/Akt/mTOR-IN-2 is a PI3K/AKT/mTOR pathway inhibitor.



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