About 11 results found for searched term "Mps1-IN-1" (0.239 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M13695 | Mps1-IN-1 | Others |
| Mps1-IN-1 is a potent, selective and ATP-competitive Mps1 kinase inhibitor, with an IC50 and a Kd of 367 nM and 27 nM. | ||
| M6078 | CFI-402257 | Others |
| CFI-402257 is a highly selective and orally bioavailable TTK and Mps1 inhibitor with Kis of 0.1 and 0.09 nM, respectively. | ||
| M8519 | Mps1-IN-2 | PLK |
| Mps1-IN-2 is a potent and selective inhibitor of Mps1 kinase. | ||
| M8918 | BAY 1217389 | Kinesin |
| BAY 1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM. | ||
| M8983 | Compstatin | Complement System |
| ICVVQDWGHHRCT | ||
| Compstatinis is a 13-residue cyclic peptide, binds to complement component C3 and inhibits complement activation with IC50 of 12 μM. Compstatin exhibits exclusive specificity for primate C3s and does not bind either to C3s from lower mammalian species or to two structural homologs of C3, human C4 and C5. | ||
| M9648 | Empesertib | Serine/Threonine Protease |
| BAY1161909; Mps1-IN-5 | ||
| Empesertib (BAY1161909) is an orally bioavailable, selective inhibitor of the serine/threonine monopolar spindle 1 (Mps1) kinase (IC50 of < 1 nM), with potential antineoplastic activity. | ||
| M13696 | Mps1-IN-3 | Others |
| Mps1-IN-3 is a potent and selective MPS1 kinase inhibitor, with an IC50 of 50 nM. | ||
| M21002 | BOS172722 | Others |
| BOS172722 is a monopolar spindle 1 (MPS1) checkpoint inhibitor with IC50 of 11 nM, Ki of 0.11 nM. | ||
| M29751 | RMS-07 | Mps1/TTK |
| RMS-07 is a covalent Monopolar Spindle Kinase 1 (MPS1/TTK) inhibitor, with an apparent IC50 of 13.1 nM. RMS-07 targets a poorly conserved cysteine in the kinase's hinge region. | ||
| M41545 | Mps1-IN-6 | Mps1/TTK |
| Mps1-IN-6 is a potent Mps1 inhibitor with an IC50 value of 2.596 nM. | ||
| M56001 | Luvixasertib hydrochloride | Mps1/TTK |
| CFI-402257 hydrochloride is a highly selective and orally bioavailable TTK/Mps1 inhibitor with an IC50 of 1.7 nM for TTK in vitro. | ||
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