About 13 results found for searched term "CALP1" (0.497 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M28012 | Acetyl-Calpastatin(184-210)(human) | Proteasome |
| Acetyl-Calpastatin(184-210)(human) is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively. | ||
| M31060 | Acetyl-Calpastatin(184-210)(human) TFA | Proteasome |
| Acetyl-Calpastatin(184-210)(human) TFA is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively. | ||
| M51696 | Calpain-1 substrate, fluorogenic | Fluorescent Dye |
| Calpain-1 substrate, fluorogenic serves as a sensitive and specific substrate for calpain-1 that cleaves Tyr-Gly bond and results in enhanced fluorescence.(Ex/Em = 490 nm/518 nm). | ||
| M53076 | CALP1 | GluR |
| CALP1 is a calmodulin (CaM) agonist (Kd of 88 µM) with binding to the CaM EF-hand/Ca2+-binding site. | ||
| M3636 | Leupeptin hemisulfate | Cathepsin |
| Leupeptin hemisulfate hemisulfate is the reversible inhibitor of lysosomal serine and cysteine proteinases; Leupeptin; inhibition of cathepsin B(Ki=6 nM), calpain(Ki=10 nM), trypsin (Ki=35 nM), plasmin (Ki=3.4 μM) and kallikrein (Ki=19 μM) had no effect on chymotrypsin, elastase, renin, or pepsin. | ||
| M5221 | MG-101 | Proteasome |
| Calpain inhibitor I; Ac-LLnL-CHO; ALLN | ||
| MG-101 is a potent inhibitor of cysteine proteases including calpain I (Ki = 190 nM), calpain II (Ki = 220 nM), cathepsin B (Ki = 150 nM), and cathepsin L (Ki = 500 pM). IC50 value: 150 nM (Ki) | ||
| M7764 | PD150606 | Proteasome |
| PD150606 is a selective, cellular permeable non-peptide calpain inhibitor with Ki of 0.21 μ m and 0.37 μ m on μ-calpains and M-calpains, respectively, and has neuroprotective activity. | ||
| M7934 | MDL 28170 | Gamma-secretase/Beta-secretase |
| Calpain Inhibitor III | ||
| Mdl-28170 (Calpain Inhibitor III) is a potent, selective, membrane-permeable Inhibitor of cysteine protease (Calpain Inhibitor III) that can quickly cross the blood-brain barrier after systemic administration. Mdl-28170 also blocks gamma-secretase. | ||
| M11294 | Alicapistat | Proteasome |
| ABT-957 | ||
| Alicapistat (ABT-957) is an orally active, selective inhibitor of human calpains 1 and 2 that can be used in alzheimer's disease (AD) studies. | ||
| M13366 | (R)-MG-132 | Proteasome |
| Z-Leu-Leu-Leu-al | ||
| (R)-MG-132 (Z-LEu-LEu-Al) is a cellular permeable proteasome and Calpain inhibitor with IC50 of 100 nM and 1.2 μM, respectively. | ||
| M28912 | (Rac)-Calpain Inhibitor XII | Proteasome |
| (Rac)-Calpain Inhibitor XII is a reversible and selective inhibitor of calpain I (μ-calpain, Ki=19 nM). (Rac)-Calpain Inhibitor XII has lower affinities for calpain II (m-calpain, Ki=120 nM) and cathepsin B (Ki=750 nM). | ||
| M29365 | Dazcapistat | Proteasome |
| Dazcapistat is a potent calpain inhibitor, with IC50s of <3 μM for calpain 1, calpain 2 and calpain 9, respectively. | ||
| M58191 | Calphostin C | Wnt/beta-catenin |
| PKF115-584; UCN-1028C | ||
| Calphostin C (PKF115-584) is a small molecule inhibitor of Wnt/beta-catenin/lef-1 signaling. Calphostin C is also a potent and specific inhibitor of protein kinase C. PKF115-584 efficiently killed CLL cells (LC(50)<1 microM), whereas normal B cells were not significantly affected. | ||
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