About 11 results found for searched term "5-HT1A antagonist 1" (0.124 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M54595 | 5-HT1A antagonist 1 | 5-HT Receptor |
| 5-HT1A antagonist 1 is a potent and selective 5-HT1A receptor antagonist with a Ki value of 35 nM.5-HT1A antagonist 1 can be used in the study of central nervous system disorders. | ||
| M3481 | WAY-100635 Maleate | 5-HT Receptor |
| WAY-100635 maleate is a potent, selective 5-HT1A receptor antagonist with an IC50 value of 0.91 nM, a Ki value of 0.39 nM, and a pIC50 of 8.87, which is more than 100-fold more selective than for use at the other 5-HT receptor subtypes and major neurotransmitter receptors. In addition, WAY-100635 maleate is a potent dopamine D4 receptor agonist. | ||
| M3818 | Rotigotine Hydrochloride | Dopamine Receptor |
| Rotigotine HCl;N-0923 Hydrochloride | ||
| Rotigotine Hydrochloride (N-0923 Hydrochloride) is a full agonist of dopamine receptor, a partial agonist of the 5-HT1A receptor, and an antagonist of the α2B-adrenergic receptor, with Ki of 0.71 nM, 4-15 nM, and 83 nM for the dopamine D3 receptor and D2, D5, D4 receptors, and dopamine D1 receptor. | ||
| M13865 | Alprenolol | 5-HT Receptor |
| (RS)-Alprenolol; dl-Alprenolol | ||
| Alprenolol is a non-selective beta blocker as well as 5-HT1A receptor antagonist. The reference for administration is 10 mg/kg. | ||
| M13866 | Alprenolol hydrochloride | 5-HT Receptor |
| (RS)-Alprenolol hydrochloride; dl-Alprenolol hydrochloride | ||
| Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. The reference for administration is 10 mg/kg. | ||
| M19276 | Rotundine | 5-HT Receptor |
| (-)-Tetrahydropalmatine; L-Tetrahydropalmatine | ||
| Rotundine is an antagonist of 5-HT1A with an IC50 of 370 nM. Rotundine is also an antagonist of dopamine D1, D2 and D3 receptors with IC50s of 166 nM, 1.4 μM and 3.3 μM, respectively. | ||
| M20391 | Naftopidil DiHCl | Adrenergic Receptor |
| KT-611 | ||
| Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively. | ||
| M28018 | Brilaroxazine | Dopamine Receptor |
| RP5063 | ||
| Brilaroxazine (RP5603) is a potent and orally active multimodal dopamine (DA)/serotonin (5-HT) modulator. Brilaroxazine is a partial agonist of dopamine (DA) D2, D3, and D4 receptors, 5-HT1A (Ki=1.5 nM) and 5-HT2A (Ki=2.5 nM), and has antagonist activity at 5-HT2B (Ki=0.19 nM), and 5-HT7 (Ki=2.7 nM) receptors. | ||
| M29350 | p-MPPI hydrochloride | 5-HT Receptor |
| p-MPPI hydrochloride is a selective 5-HT1A receptor antagonist with high affinity for 5-HT1A receptors. p-MPPI hydrochloride can crosses the blood-brain barrier, and has clear antidepressant and anxiolytic-like effects. | ||
| M30957 | Piromelatine | Melatonin Receptor |
| Neu-P11 | ||
| Piromelatine (Neu-P11) is a melatonin MT1/MT2 receptor agonist, serotonin 5-HT1A/5-HT1D agonist, and serotonin 5-HT2B antagonist. Piromelatine (Neu-P11) possesses sleep promoting, analgesic, anti-neurodegenerative, anxiolytic and antidepressant potentials. Piromelatine (Neu-P11) also possesses pain-related P2X3, TRPV1, and Nav1.7 channel-inhibition capacities. | ||
| M49351 | AX-1602 | 5-HT Receptor |
| AX-1602 is a 5-HT1A receptor antagonist, adrenergic receptor ADRA2 agonist, and cannabinoid receptor CB1 antagonist for studies related to atopic dermatitis, psoriasis, and vitiligo. | ||
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