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Xanomeline

Cat. No. M10906

All AbMole products are for research use only, cannot be used for human consumption.

Xanomeline  Structure
Synonym:

LY-246708

Size Price Availability Quantity
1mg USD 30  USD30 In stock
5mg USD 55  USD55 In stock
10mg USD 95  USD95 In stock
25mg USD 185  USD185 In stock
50mg USD 300  USD300 In stock
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Quality Control & Documentation
Biological Activity

Xanomeline increases neuronal excitability as a potent selective muscarinic 1 and type 4 (M1/M4) receptor agonist. Xanomeline can be used in the study of neurological disorders such as schizophrenia.

Chemical Information
Molecular Weight 281.42
Formula C14H23N3OS
CAS Number 131986-45-3
Solubility (25°C) DMSO ≥ 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Stephen K Brannan, et al. N Engl J Med. Muscarinic Cholinergic Receptor Agonist and Peripheral Antagonist for Schizophrenia

[2] Rujuan Xin, et al. Front Physiol. Xanomeline Protects Cortical Cells From Oxygen-Glucose Deprivation via Inhibiting Oxidative Stress and Apoptosis

[3] Aaron M Bender, et al. ACS Chem Neurosci. Classics in Chemical Neuroscience: Xanomeline

[4] Naheed R Mirza, et al. CNS Drug Rev. Xanomeline and the antipsychotic potential of muscarinic receptor subtype selective agonists

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Keywords: Xanomeline , LY-246708 supplier, AChR/AChE, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



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