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Ensartinib

Cat. No. M28270

All AbMole products are for research use only, cannot be used for human consumption.

Ensartinib Structure
Synonym:

X-396

Size Price Availability Quantity
1mg USD 60  USD60 In stock
5mg USD 140  USD140 In stock
10mg USD 220  USD220 In stock
25mg USD 460  USD460 In stock
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Quality Control & Documentation
Biological Activity

Ensartinib (X-396) is a potent and dual ALK/MET inhibitor with IC50s of <0.4 nM and 0.74 nM, respectively.

Chemical Information
Molecular Weight 561.44
Formula C26H27Cl2FN6O3
CAS Number 1370651-20-9
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Yuxiang Ma, et al. J Thorac Dis. Ensartinib in advanced ALK-positive non-small cell lung cancer: a multicenter, open-label, two-staged, phase 1 trial

[2] Yunpeng Yang, et al. Lancet Respir Med. Efficacy, safety, and biomarker analysis of ensartinib in crizotinib-resistant, ALK-positive non-small-cell lung cancer: a multicentre, phase 2 trial

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  Catalog
Abmole Inhibitor Catalog




Keywords: Ensartinib, X-396 supplier, ALK, inhibitors, activators

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