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WH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6 nM. WH-4-023 has little inhibition on p38α and KDR.
| Molecular Weight | 568.67 |
| Formula | C32H36N6O4 |
| CAS Number | 837422-57-8 |
| Solubility (25°C) | DMSO 15 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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