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Valecobulin

Cat. No. M27906

All AbMole products are for research use only, cannot be used for human consumption.

Valecobulin Structure
Synonym:

CKD-516

Price and Availability

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Quality Control & Documentation
Biological Activity

Valecobulin (CKD516) is a valine proagent of (S516) and a vascular disrupting agent (VDA). Valecobulin is a potent β-tubulin polymerization inhibitor with marked antitumor activity against murine and human solid tumors.

Chemical Information
Molecular Weight 536.6
Formula C26H28N6O5S
CAS Number 1188371-47-2
Form Solid
Solubility (25°C) DMSO 125 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Soo Jin Kim, et al. Cancer Chemother Pharmacol. Involvement of ER stress and reactive oxygen species generation in anti-cancer effect of CKD-516 for lung cancer

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Keywords: Valecobulin, CKD-516 supplier, Microtubule, inhibitors, activators

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