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U7D-1 is a first-in-class, potent and selective ubiquitin-specific protease 7 USP7 PROTAC depressant in RS4; The DC50 in 11 cells was 33 nM. U7D-1 has anti-cancer activity.
| Molecular Weight | 940.14 |
| Formula | C53H65N9O7 |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Yuan Pei, et al. Angew Chem Int Ed Engl. Discovery of a Potent and Selective Degrader for USP7
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