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TP0597850 

Cat. No. M29749

All AbMole products are for research use only, cannot be used for human consumption.

TP0597850  Structure

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Quality Control & Documentation
Biological Activity

TP0597850 is a selective inhibitor of MMP2 (IC50=0.22 nM). TP0597850 has a long MMP2 dissociation half-life (t1/2=265 min).

Chemical Information
Molecular Weight 916.01
Formula C41H57N9O13S
CAS Number 2642181-22-2
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Tomoki Takeuchi, et al. J Med Chem. Discovery of TP0597850: A Selective, Chemically Stable, and Slow Tight-Binding Matrix Metalloproteinase-2 Inhibitor with a Phenylbenzamide-Pentapeptide Hybrid Scaffold

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  Catalog
Abmole Inhibitor Catalog




Keywords: TP0597850  supplier, MMP, inhibitors, activators

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