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THRX-160209

Cat. No. M54823

All AbMole products are for research use only, cannot be used for human consumption.

THRX-160209 Structure
Synonym:

THRX160209

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Quality Control & Documentation
Biological Activity

THRX-160209 is a potent antagonist at the M(2) muscarinic acetylcholine (ACh) receptor subtype that was designed using a multivalent strategy, simultaneously targeting the orthosteric site and a nearby site known to bind allosteric ligands.

Chemical Information
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Tod Steinfeld, et al. Mol Pharmacol. A novel multivalent ligand that bridges the allosteric and orthosteric binding sites of the M2 muscarinic receptor

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Keywords: THRX-160209, THRX160209 supplier, AChR/AChE, inhibitors, activators

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