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TC-E 5001 

Cat. No. M30744

All AbMole products are for research use only, cannot be used for human consumption.

TC-E 5001  Structure

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Quality Control & Documentation
Biological Activity

TC-E 5001 is an inhibitor of Wnt pathway that inhibits tankyrase 1/2 (TNKS1/2) via novel adenosine pocket binding, with Kds of 79 nM and 28 nM, respectively. TC-E 5001 also inhibits Axin2 and STF, with IC50s of 0.709 μM and 0.215 μM, respectively.

Chemical Information
Molecular Weight 409.46
Formula C20H19N5O3S
CAS Number 865565-29-3
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Vegard Torp Lien, et al. RSC Adv. Towards dual inhibitors of the MET kinase and WNT signaling pathway; design, synthesis and biological evaluation

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  Catalog
Abmole Inhibitor Catalog




Keywords: TC-E 5001  supplier, PARP, inhibitors, activators

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