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Osavampator (TAK-653) is a potential first-in-class alpha amino-3-hydroxy-5-methyl-4-isoxazole propionic acid (AMPA) enhancer. Osavampator selectively binds to AMPA-R in a glutamate-dependent manner and induces Ca2+ influx in hGluA1i CHO cells (EC50 = 3.3 μM).
| Molecular Weight | 373.47 |
| Formula | C19H23N3O3S |
| CAS Number | 1358751-06-0 |
| Form | Solid |
| Solubility (25°C) | DMSO 10 mg/mL |
| Storage | 2-8°C, protect from light, dry, sealed |
[5] Jeffrey M Witkin, et al. Adv Pharmacol. Rapid-acting antidepressants
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