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SZUH280 is a potent and selective PROTAC HDAC8 degrader with a DC50 of 0.58 μM in A549 cells. SZUH280 induces cancer cell apoptosis. SZUH280 hampers DNA damage repair in cancer cells, promoting cellular radiosensitization.
| Molecular Weight | 706.7 |
| Formula | C36H34N8O8 |
| CAS Number | 2770263-77-7 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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