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SJ10542 is a potent and selective JAK2/3 directing phenyl glutarimide (PG)-PROTAC with DC50s of 14, 11, and 24 nM for JAK2, JAK3, and JAK2-fusion ALL, respectively.
| Molecular Weight | 818.95 |
| Formula | C41H46N12O5S |
| CAS Number | 2789678-92-6 |
| Form | Solid |
| Solubility (25°C) | DMSO 40 mg/mL (ultrasonic) |
| Storage | 4°C, dry, sealed |
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