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Sepimostat (FUT-187 free base) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat inhibits the Ifenprodil binding with a Ki value of 27.7 µM.
| Molecular Weight | 373.41 |
| Formula | C21H19N5O2 |
| CAS Number | 103926-64-3 |
| Form | Solid |
| Solubility (25°C) | DMSO 6.25 mg/mL (ultrasonic) |
| Storage | Powder -20°C |
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