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SAR629 

Cat. No. M27967

All AbMole products are for research use only, cannot be used for human consumption.

SAR629  Structure

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Quality Control & Documentation
Biological Activity

SAR629 is a potent monoglyceride lipase (MGL) covalent inhibitor. SAR629 also inhibits 2-Arachidonoylglycerol (2-AG) degradation.

Chemical Information
Molecular Weight 383.39
Formula C20H19F2N5O
CAS Number 1221418-42-3
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Francesca Galvani, et al. J Chem Inf Model. Mechanistic Modeling of Monoglyceride Lipase Covalent Modification Elucidates the Role of Leaving Group Expulsion and Discriminates Inhibitors with High and Low Potency

[2] T Bertrand, et al. J Mol Biol. Structural basis for human monoglyceride lipase inhibition

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  Catalog
Abmole Inhibitor Catalog




Keywords: SAR629  supplier, MAGL, inhibitors, activators

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