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Rodatristat (KAR5417) is a potent tryptophan hydroxylase 1 (TPH1) and TPH2 inhibitor with IC50s value of 33 nM and 7 nM, respectively, and shows robust reduction of intestinal serotonin (5-HT) levels in mice.
| Molecular Weight | 561.98 |
| Formula | C27H27ClF3N5O3 |
| CAS Number | 1673568-73-4 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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