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Rivanicline hemioxalate

Cat. No. M31050

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Rivanicline hemioxalate Structure
Synonym:

RJR-2403 hemioxalate; (E)-Metanicotine hemioxalate

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Quality Control & Documentation
Biological Activity

Rivanicline hemioxalate (RJR-2403 hemioxalate; (E)-Metanicotine hemioxalate) is a neuronal nicotinic receptor agonist, showing high selectivity for the α4β2 subtype (Ki=26 nM); > 1,000 fold selectivity than α7 receptors(Ki= 3.6 μM).

Chemical Information
Molecular Weight 207.23
Formula C11H15N2O2
Form Solid
Solubility (25°C) DMSO 50 mg/mL (ultrasonic)
Storage 4°C, dry, sealed
References

[1] Marieta Muresan-Pop, et al. Acta Crystallogr C Struct Chem. New solvates and a salt of the anti-HIV compound etravirine

[2] Lamia Bendjeddou, et al. Acta Crystallogr Sect E Struct Rep Online. 3-Carboxy-anilinium hemioxalate

[3] Zhan Tang, et al. Acta Crystallogr Sect E Struct Rep Online. N-[2-(2-Chloro-phen-yl)-2-hydroxy-ethyl]propan-2-aminium hemioxalate

[4] Leila Narimani, et al. Acta Crystallogr Sect E Struct Rep Online. Ethyl-enediaminium hemioxalate thio-cyanate

[5] B Sridhar, et al. Acta Crystallogr C. Multicomponent crystals of erlotinib

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Keywords: Rivanicline hemioxalate, RJR-2403 hemioxalate; (E)-Metanicotine hemioxalate supplier, AChR/AChE, inhibitors, activators

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