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Risperidone hydrochloride

Cat. No. M30448

All AbMole products are for research use only, cannot be used for human consumption.

Risperidone hydrochloride Structure
Synonym:

R 64 766 hydrochloride

Price and Availability

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Quality Control & Documentation
Biological Activity

Risperidone hydrochloride (R 64 766 hydrochloride) 5-HT2 receptor blocker, P-Glycoprotein inhibitor and potent dopamine D2 receptor antagonist, with Kis of 4.8, 5.9 nM for 5-HT2A and dopamine D2 receptor, respectively.

Chemical Information
Molecular Weight 446.95
Formula C23H28ClFN4O2
CAS Number 666179-74-4
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Filip Milosavljevic, et al. JAMA Psychiatry. Association of CYP2C19 and CYP2D6 Poor and Intermediate Metabolizer Status With Antidepressant and Antipsychotic Exposure: A Systematic Review and Meta-analysis

[2] Stefan Leucht, et al. Am J Psychiatry. Dose-Response Meta-Analysis of Antipsychotic Drugs for Acute Schizophrenia

[3] Yi-Cheng Wu, et al. JAMA Psychiatry. Association of Delirium Response and Safety of Pharmacological Interventions for the Management and Prevention of Delirium: A Network Meta-analysis

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  Catalog
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Keywords: Risperidone hydrochloride, R 64 766 hydrochloride supplier, 5-HT Receptor, inhibitors, activators

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