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Remogliflozin etabonate (GSK189075)

Cat. No. M20997

All AbMole products are for research use only, cannot be used for human consumption.

Remogliflozin etabonate (GSK189075) Structure

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Quality Control & Documentation
Biological Activity

Remogliflozin etabonate (GSK189075) is an orally active, selective and low-affinity inhibitor of sodium glucose cotransporter (SGLT2) with Ki of 1950 nM, 2140 nM, 43100 nM, 8570 nM for hSGLT2, rSGLT2, hSGLT1, rSGLT1, respectively. Remogliflozin etabonate exhibits antidiabetic efficacy in rodent models.

Chemical Information
Molecular Weight 522.59
Formula C26H38N2O9
CAS Number 442201-24-3
Solubility (25°C) DMSO 100 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Robert Dobbins, et al. BMC Pharmacol Toxicol. Assessment of safety and tolerability of remogliflozin etabonate (GSK189075) when administered with total daily dose of 2000 mg of metformin

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  Catalog
Abmole Inhibitor Catalog




Keywords: Remogliflozin etabonate (GSK189075) supplier, SGLT, inhibitors, activators

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