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(Rac)-PF-4136309 is an isoform of PF-4136309. PF-4136309 (INCB8761, PF-04136309) is a potent, selective, and orally bioavailable CCR2 antagonist with an IC50 of 5.2 nM for human CCR2.
| Molecular Weight | 568.59 |
| Formula | C29H31F3N6O3 |
| CAS Number | 857679-55-1 |
| Solubility (25°C) | DMSO 30 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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