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Progabide

Cat. No. M31352

All AbMole products are for research use only, cannot be used for human consumption.

Progabide Structure
Synonym:

SL 76002

Price and Availability

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Quality Control & Documentation
Biological Activity

Progabide is a gamma-aminobutyric acid (GABA) receptor agonist that may be used in studies related to epilepsy.

Chemical Information
Molecular Weight 334.77
Formula C17H16ClFN2O2
CAS Number 62666-20-0
Form Solid
Solubility (25°C) DMSO >100 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] C Cepeda, et al. Epilepsia. Action of progabide in the photosensitive baboon, Papio papio

[2] J M Martínez-Lage, et al. Epilepsia. Progabide treatment in severe epilepsy: a double-blind cross-over trial versus placebo

[3] H Manev, et al. Pharmacol Biochem Behav. Progabide, a GABA mimetic drug, stimulates the secretion of plasma corticosterone in rats

[4] G H Fromm, et al. Epilepsia. Comparison of progabide with other antiepileptic and GABAergic drugs

[5] K J Bergmann. Clin Neuropharmacol. Progabide: a new GABA-mimetic agent in clinical use

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Keywords: Progabide, SL 76002 supplier, GABA Receptor, inhibitors, activators

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