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Picfeltarraegenin X

Cat. No. M10655
Picfeltarraegenin X Structure
Synonym:

Picfeltarraenin X

Size Price Availability Quantity
2mg USD 270  USD270 In stock
5mg USD 490  USD490 In stock
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Quality Control & Documentation
Biological Activity

Picfeltarraenin X is an AChE inhibitor, which is a triterpenoid isolated from Picria fel-terrae Lour.

Chemical Information
Molecular Weight 662.81
Formula C36H54O11
CAS Number 1391826-61-1
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Conversion of different model animals based on BSA (PMID: 27057123)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of Compound A used for a mouse (20 mg/kg) to a dose based on the BSA for a rat, multiply 20 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for Compound A of 10 mg/kg.

References

[1] L-Sheng Wang, et al. J Asian Nat Prod Res. Two new triterpenoids from Picria fel-terrae

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Keywords: Picfeltarraegenin X, Picfeltarraenin X supplier, AChR/AChE, inhibitors, activators


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