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Perospirone (SM-9018 free base) is an orally active antagonist of 5-hydroxytryptamine2 (5-HT2) receptor, dopamine2 (D2) receptor and 5-HT1A receptor with Ki of 0.6 nM, 1.4 nM and 2.9 nM, respectively.
| Molecular Weight | 426.57 |
| Formula | C23H30N4O2S |
| CAS Number | 150915-41-6 |
| Solubility (25°C) | DMSO 85 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] Tomas de Paulis. Curr Opin Investig Drugs. Perospirone (Sumitomo Pharmaceuticals)
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