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PB131

Cat. No. M41490

All AbMole products are for research use only, cannot be used for human consumption.

PB131 Structure

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Quality Control & Documentation
Biological Activity

PB131 is a selective and brain-permeable HDAC6 inhibitor with high binding affinity (IC50: 1.8 nM).

Chemical Information
Molecular Weight 301.32
Formula C16H16FN3O2
CAS Number 2924425-63-6
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Gang Liu et al. Eur J Med Chem. Design, synthesis, and anti-inflammatory activity characterization of novel brain-permeable HDAC6 inhibitors

[2] Hélène Brodeur et al. Biochem Cell Biol. Kinetic properties of chimeric class I aldehyde dehydrogenases for retinal isomers

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  Catalog
Abmole Inhibitor Catalog




Keywords: PB131 supplier, HDAC, inhibitors, activators

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