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Palonosetron

Cat. No. M20533

All AbMole products are for research use only, cannot be used for human consumption.

Palonosetron Structure
Synonym:

RS25259, RS 25259 197

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Quality Control & Documentation
Biological Activity

Palonosetron is a 5-HT3 antagonist with a Ki value of 0.17 nM and may be used in studies related to nausea and vomiting.

Chemical Information
Molecular Weight 296.41
Formula C19H24N2O
CAS Number 135729-61-2
Solubility (25°C) DMSO 59 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Matti Aapro, et al. Curr Cancer Drug Targets. Netupitant-palonosetron (NEPA) for Preventing Chemotherapy-induced Nausea and Vomiting: From Clinical Trials to Daily Practice

[2] No authors listed. Palonosetron

[3] Rudolph M Navari. Expert Opin Pharmacother. Palonosetron for the treatment of chemotherapy-induced nausea and vomiting

[4] Lily P H Yang, et al. Drugs. Palonosetron: in the prevention of nausea and vomiting

[5] M Asif A Siddiqui, et al. Drugs. Palonosetron

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  Catalog
Abmole Inhibitor Catalog




Keywords: Palonosetron, RS25259, RS 25259 197 supplier, 5-HT Receptor, inhibitors, activators

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