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Ocaperidone

Cat. No. M13872

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Ocaperidone Structure
Synonym:

R79598

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Biological Activity

Ocaperidone is an effective antipsychotic agent, acting as a potent 5-HT2 and dopamine D2 antagonist, and a 5-HT1A agonist, with Kis of 0.14 nM, 0.46 nM, 0.75 nM, 1.6 nM and 5.4 nM for 5-HT2, a1-adrenergic receptor, dopamine D2, histamine H1 and a2-adrenergic receptor, respectively, and a pEC50 and pKi of 7.60 and 8.08 for h5-HT1A.

Chemical Information
Molecular Weight 420.48
CAS Number 129029-23-8
Solubility (25°C) DMSO 16.67 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hugo Geerts, et al. Blinded prospective evaluation of computer-based mechanistic schizophrenia disease model for predicting drug response

[2] R Brys, et al. Reconstitution of the human 5-HT(1D) receptor-G-protein coupling: evidence for constitutive activity and multiple receptor conformations

[3] J E Leysen, et al. In vitro and in vivo receptor binding and effects on monoamine turnover in rat brain regions of the novel antipsychotics risperidone and ocaperidone

[4] A A Megens, et al. Behavioral disinhibition and depression in amphetaminized rats: a comparison of risperidone, ocaperidone and haloperidol

[5] A A Megens, et al. Pharmacological profile of the new potent neuroleptic ocaperidone (R 79,598)

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Keywords: Ocaperidone, R79598 supplier, 5-HT Receptor, inhibitors, activators

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