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Norfluoxetine hydrochloride

Cat. No. M7799

All AbMole products are for research use only, cannot be used for human consumption.

Norfluoxetine hydrochloride Structure
Size Price Availability Quantity
2mg USD 75  USD75 In stock
5mg USD 120  USD120 In stock
10mg USD 175  USD175 In stock
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Quality Control & Documentation
Biological Activity

Norfluoxetine hydrochloride is an active N-demethylated fluoxetine metabolite, Norfluoxetine hydrochloride is more potent inhibitor of serotonin uptake than fluoxetine with a half-life in vivo of 5-7 days.

Chemical Information
Molecular Weight 331.76
Formula C16H16F3NO · HCl
CAS Number 57226-68-3
Solubility (25°C) Water 4 mg/mL
DMSO 60 mg/mL
Storage 4°C, dry, sealed
References

[1] Hyeon-Cheol Jeong, et al. Prediction of Fluoxetine and Norfluoxetine Pharmacokinetic Profiles Using Physiologically Based Pharmacokinetic Modeling

[2] No authors listed. Fluoxetine

[3] C Hiemke, et al. Pharmacokinetics of selective serotonin reuptake inhibitors

[4] R C Pohland, et al. Postmortem serum and tissue redistribution of fluoxetine and norfluoxetine in dogs following oral administration of fluoxetine hydrochloride (Prozac)

[5] A C Altamura, et al. Clinical pharmacokinetics of fluoxetine

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