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MSC-4106

Cat. No. M31170

All AbMole products are for research use only, cannot be used for human consumption.

MSC-4106 Structure

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Quality Control & Documentation
Biological Activity

MSC-4106 is an orally active inhibitor of the YAP/TAZ-TEAD complex that blocks the auto-palmitoylation of TEAD1 and TEAD3, and can be used for tumor-related studies.

Chemical Information
Molecular Weight 359.3
Formula C18H12F3N3O2
CAS Number 2738542-58-8
Form Solid
Solubility (25°C) DMSO >100 mg/mL
Storage -20°C, dry, sealed
References

[1] Timo Heinrich, et al. J Med Chem. Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106

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  Catalog
Abmole Inhibitor Catalog




Keywords: MSC-4106 supplier, YAP, inhibitors, activators

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