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MK-8153

Cat. No. M21142

All AbMole products are for research use only, cannot be used for human consumption.

MK-8153  Structure

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Quality Control & Documentation
Biological Activity

MK-8153 is a potent, selective and orally active extrarenal medullary potassium channel (ROMK) inhibitor with IC50 values of 5 nM and 34 μM for ROMK EP and hERG EP, respectively.MK-8153 can be used as a diuretic.

Chemical Information
Molecular Weight 440.49
Formula C24H28N2O6
CAS Number 1548286-45-8
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jinlong Jiang, et al. J Med Chem. Discovery of MK-8153, a Potent and Selective ROMK Inhibitor and Novel Diuretic/Natriuretic

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  Catalog
Abmole Inhibitor Catalog




Keywords: MK-8153 supplier, Potassium Channel, inhibitors, activators

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