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MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1, with an IC50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4.0 nM in IMR-32 cells.
| Molecular Weight | 424.42 |
| Formula | C23H21FN2O5 |
| CAS Number | 863115-70-2 |
| Form | Solid |
| Solubility (25°C) | DMSO 10 mg/mL (ultrasonic and adjust pH to 6 with HCl) |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] Anders Johansson, et al. Expert Opin Ther Pat. Novel MCH1 receptor antagonists: a patent review
[3] Denise Andersen, et al. J Org Chem. Stereoselective synthesis of a MCHr1 antagonist
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