Certificate of Analysis
| Product Name: | MCHR1 antagonist 2 |
| Catalog Number: | M30725 |
| CAS Number: | 863115-70-2 |
Physical and Chemical Properties
| Formula: | C23H21FN2O5 |
| Molecular Weight: | 424.42 |
| Form: | Solid |
| Solubility: | DMSO 10 mg/mL (ultrasonic and adjust pH to 6 with HCl) |
| Storage: |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Chemical Structure: |  |
Analytical Data
| QC Standard: | ≥99.0% |
| H-NMR: | Consistent with structure |
Product Information
| Description: | MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1, with an IC50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4.0 nM in IMR-32 cells. |
| Stability and Solubility Advice: | Information concerning product stability, particularly in solution, has rarely been reported and in most cases we can only offer a general guide. We recommend that stock solutions, once prepared, are stored aliquoted in tightly sealed vials and used within 1 month. Avoid repeated freeze and thaw cycles. Storage conditions for some special products should refer to their storage details. |