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Lurasidone

Cat. No. M13870

All AbMole products are for research use only, cannot be used for human consumption.

Lurasidone Structure
Synonym:

SM-13496

Size Price Availability Quantity
10mg USD 50  USD50 In stock
50mg USD 130  USD130 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7 with IC50s of 1.68 and 0.495 nM, respectively. Lurasidone (SM-13496) is also a partial agonist of 5-HT1A receptor with an IC50 of 6.75 nM.

*The compound is unstable in solutions, freshly prepared is recommended



Chemical Information
Molecular Weight 492.68
CAS Number 367514-87-2
Solubility (25°C) DMSO 20.83 mg/mL
Storage 2-8°C, protect from light
References

[1] Herbert Y Meltzer, et al. Lurasidone Improves Psychopathology and Cognition in Treatment-Resistant Schizophrenia

[2] No authors listed. Lurasidone

[3] No authors listed. Lurasidone

[4] Filippo Corponi, et al. Novel antipsychotics specificity profile: A clinically oriented review of lurasidone, brexpiprazole, cariprazine and lumateperone

[5] Yusra Azhar, et al. Lurasidone

[6] No authors listed. Lurasidone

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  Catalog
Abmole Inhibitor Catalog




Keywords: Lurasidone, SM-13496 supplier, 5-HT Receptor, inhibitors, activators

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