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Lurasidone hydrochloride

Cat. No. M2825

All AbMole products are for research use only, cannot be used for human consumption.

Lurasidone hydrochloride Structure
Synonym:

SM-13496

Size Price Availability Quantity
10mg USD 40  USD40 In stock
50mg USD 110  USD110 In stock
100mg USD 170  USD170 In stock
200mg USD 270  USD270 In stock
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Quality Control & Documentation
Biological Activity

Lurasidone is an atypical antipsychotic, inhibits Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C with IC50 of 1.68 nM, 2.03 nM, 0.495 nM, 6.75 nM and 10.8 nM, respectively.

Chemical Information
Molecular Weight 529.14
Formula C28H36N4O2S.HCl
CAS Number 367514-88-3
Solubility (25°C) DMSO 1 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Khai Tran, et al. Lurasidone Hydrochloride for Bipolar Disorder: A Review of Clinical Effectiveness, Cost-Effectiveness, and Guidelines [Internet]

[2] Herbert Y Meltzer, et al. Lurasidone Improves Psychopathology and Cognition in Treatment-Resistant Schizophrenia

[3] Filippo Corponi, et al. Novel antipsychotics specificity profile: A clinically oriented review of lurasidone, brexpiprazole, cariprazine and lumateperone

[4] Michele Fornaro, et al. Lurasidone in the Treatment of Bipolar Depression: Systematic Review of Systematic Reviews

[5] No authors listed. Lurasidone Hydrochloride (Latuda): Management of Manifestations of Schizophrenia [Internet]

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Keywords: Lurasidone hydrochloride, SM-13496 supplier, 5-HT Receptor, inhibitors, activators

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