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Levomepromazine (Methotrimeprazine) is an orally available neuroleptic agent, which is commonly used to relieve nausea and vomiting in palliative care settings. Levomepromazine has antagonist actions at multiple neurotransmitter receptor sites, including dopaminergic, cholinergic, serotonin and histamine receptors.
| Molecular Weight | 328.47 |
| Formula | C19H24N2OS |
| CAS Number | 60-99-1 |
| Form | Solid |
| Solubility (25°C) | DMSO 41.67 mg/mL (ultrasonic and warming and heat to 60°C) |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] Parthipan Sivaraman, et al. Schizophr Bull. Levomepromazine for schizophrenia
[4] Parthipan Sivaraman, et al. Cochrane Database Syst Rev. Levomepromazine for schizophrenia
[5] Ben Green, et al. Curr Med Res Opin. Focus on levomepromazine
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