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Lapatinib ditosylate (GW572016 ditosylate) is a potent inhibitor of the ErbB-2 and EGFR tyrosine kinase domains with IC50 values against purified EGFR and ErbB-2 of 10.2 and 9.8 nM, respectively.
| Molecular Weight | 925.46 |
| Formula | C43H42ClFN4O10S3 |
| CAS Number | 388082-77-7 |
| Solubility (25°C) | DMSO 100 mg/mL |
| Storage | 2-8°C, protect from light, dry, sealed |
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