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L-778123 hydrochloride

Cat. No. M5024

All AbMole products are for research use only, cannot be used for human consumption.

L-778123 hydrochloride Structure
Synonym:

L-778,123 hydrochloride

Size Price Availability Quantity
1mg USD 50  USD50 In stock
5mg USD 75  USD75 In stock
10mg USD 110  USD110 In stock
50mg USD 315  USD315 In stock
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Quality Control & Documentation
Biological Activity

L-778123 hydrochloride is a dual inhibitor of FPTase and GGptase-I with IC50 values of 2 nM and 98 nM, respectively.

Chemical Information
Molecular Weight 442.34
Formula C22H21Cl2N5O
CAS Number 253863-00-2
Form Solid
Solubility (25°C) DMSO:25mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Lobell RB,et.al. Mol Cancer Ther. Preclinical and clinical pharmacodynamic assessment of L-778,123, a dual inhibitor of farnesyl:protein transferase and geranylgeranyl:protein transferase type-I.

[2] Blood.

[3]

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Keywords: L-778123 hydrochloride, L-778,123 hydrochloride supplier, Farnesyl Transferase, inhibitors, activators

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