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Kx1-004 is an effective small molecule inhibitor of SRC-PTK and can be used as a potential protective compound of NIHL. Kx1-004 was further evaluated by repeated exposure at different doses, also in place of pulsed noise exposure.
Molecular Weight | 284.29 |
Formula | C16H13FN2O2 |
CAS Number | 518058-84-9 |
Form | Solid |
Solubility (25°C) | DMSO |
Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Harris KC, et al. Hear Res. Prevention of noise-induced hearing loss with Src-PTK inhibitors.
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