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Ipsapirone (TVX Q 7821) is a partial agonist of 5-HT1A receptor and also shows antagonism to 5-HT1A receptor. It also showed inhibition of 5-HT2 and α 1-adrenergic activity only at high doses.
| Molecular Weight | 401.48 |
| Formula | C19H23N5O3S |
| CAS Number | 95847-70-4 |
| Form | Solid |
| Solubility (25°C) | DMSO |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[4] R J Fanelli, et al. Ipsapirone: a novel anxiolytic and selective 5-HT1A receptor ligand
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