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INCB059872 is a potent, orally active, selective and irreversible inhibitor of lysine-specific demethylase 1 (LSD1) in myeloid leukemia.
Molecular Weight | 386.53 |
Formula | C23H34N2O3 |
CAS Number | 1802909-49-4 |
Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] Chaofeng Zhang, et al. Bioorg Chem. Recent advances of LSD1/KDM1A inhibitors for disease therapy
[5] Xiaoli Fu, et al. Future Med Chem. Advances toward LSD1 inhibitors for cancer therapy
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