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Imperatorin is a potent NO synthesis inhibitor with an IC50 of 9.2 μmol and a BChE inhibitor with an IC50 of 31.4 μmol. Imperatorin is a weak agonist of TRPV1 with an EC50 of 12.6±3.2 μM.
| Molecular Weight | 270.28 |
| Formula | C16H14O4 |
| CAS Number | 482-44-0 |
| Solubility (25°C) | DMSO ≥ 40 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] Mao Deng, et al. Imperatorin: A review of its pharmacology, toxicity and pharmacokinetics
[4] M I Nasser, et al. Effects of imperatorin in the cardiovascular system and cancer
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