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Granisetron

Cat. No. M20451

All AbMole products are for research use only, cannot be used for human consumption.

Granisetron Structure
Synonym:

Sancuso, Kevatril, Granisetronum, Sustol

Size Price Availability Quantity
25mg USD 48  USD48 In stock
50mg USD 75  USD75 In stock
100mg USD 110  USD110 In stock
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Quality Control & Documentation
Biological Activity

Granisetron is a serotonin receptor (5HT-3 selective) antagonist that is used as an antiemetic and antinauseant for cancer chemotherapy.

Chemical Information
Molecular Weight 312.41
Formula C18H24N4O
CAS Number 109889-09-0
Solubility (25°C) DMSO 11 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Mehmet Aksoy, et al. J Clin Anesth. Granisetron or ondansentron to prevent hypotension after spinal anesthesia for elective cesarean delivery: A randomized placebo-controlled trial

[2] Sheila A Doggrell. Expert Opin Pharmacother. Granisetron in the treatment of chemotherapy-induced nausea and vomiting (CINV) - is there still a role after comparison with palonosetron?

[3] Emma D Deeks. Drugs. Granisetron Extended-Release Injection: A Review in Chemotherapy-Induced Nausea and Vomiting

[4] Sean T Duggan, et al. Drugs. Transdermal granisetron

[5] M Nodoushani. Conn Med. Granisetron

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Keywords: Granisetron, Sancuso, Kevatril, Granisetronum, Sustol supplier, 5-HT Receptor, inhibitors, activators

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